PTPN11
Overview
PTPN11 (SHP2) is a tyrosine phosphatase that acts upstream of RAS/MAPK signaling. In the corpus it is a rare RAS-pathway driver in histiocytosis.
Alterations observed in the corpus
- Mutated in one histiocytosis patient in the Make-an-IMPACT rare-cancer cohort; patient was treated with a MEK inhibitor PMID:36862133.
- Activating missense mutations in 2.9% (7/240) of high-risk neuroblastomas (nbl_broad_2013); all previously reported in COSMIC; one of only 5 statistically and biologically significant recurrently mutated genes in this low-mutation-burden pediatric tumor PMID:23334666
- Activating mutations (e.g., p.Gly503Arg) found in near haploid ALL as part of RTK/Ras pathway alterations (71% of near haploid cases); one PTPN11 variant was inherited and Noonan syndrome-associated (all_stjude_2013, 124 pediatric cases) PMID:23334668
- Part of the activated-signaling gene category in AML (alongside KIT, KRAS, NRAS, FLT3); contributes to the 59% signaling-pathway prevalence across 200 AML cases PMID:23634996
- E69K and E76A activating mutations (previously described in juvenile myelomonocytic leukemia) exclusively co-occurring with FGFR1 mutations in pilocytic astrocytoma; PTPN11/SHP-2 expression globally elevated in this tumor type PMID:23817572
- 2 expressed mutations detected in rhabdomyosarcoma, both restricted to fusion-negative (PFN) tumors; PTPN11 (SHP2) encodes an RAS-activating phosphatase PMID:24436047
- Non-passenger mutation in breast adenoid cystic carcinoma (AdCC); rarely mutated in basal-like breast cancers. PMID:26095796
- E76A/K hotspot in 2 desmoplastic melanoma tumors. PMID:26343386
- Recurrent missense mutations in CLL (n=7, 1.3%); identified as a novel CLL driver modulating MYC activity in a 538-patient WES study PMID:26466571
- PTPN11 co-occurs with NPM1 and modifies outcome in NPM1-mutated AML; part of the RTK-RAS pathway group identified in a 1540-patient AML genomic study PMID:27276561.
- G503V mutation in AML (MEK-inhibitor target); D61Y co-mutation with SETBP1 D868N reclassified a 4-year-old’s diagnosis from de novo AML to JMML (which evolved into AML) in a pediatric precision-oncology cohort PMID:28007021
Cancer types (linked)
- Histiocytosis (LCH, ECD) — rare actionable alteration PMID:36862133.
Co-occurrence and mutual exclusivity
- None reported.
Therapeutic relevance
- MEK inhibitor treatment reported for PTPN11-mutant histiocytosis patient in the direct-to-patient program PMID:36862133.
Open questions
- None specific to PTPN11 in this cohort.
Sources
This page was processed by crosslinker on 2026-05-14. - PMID:23334666
This page was processed by crosslinker on 2026-05-14. - PMID:23334668
This page was processed by crosslinker on 2026-05-14. - PMID:23634996
This page was processed by crosslinker on 2026-05-14. - PMID:23817572
This page was processed by crosslinker on 2026-05-14. - PMID:24436047
This page was processed by crosslinker on 2026-05-14. - PMID:26095796
This page was processed by crosslinker on 2026-05-14. - PMID:26343386
This page was processed by crosslinker on 2026-05-14. - PMID:26466571
This page was processed by crosslinker on 2026-05-14. - PMID:27276561
This page was processed by entity-page-writer on 2026-05-15. - PMID:28007021
This page was processed by wiki-cli on 2026-05-14.