SUZ12

Overview

SUZ12 encodes a core component of the Polycomb Repressive Complex 2 (PRC2), which catalyzes histone H3 lysine 27 trimethylation (H3K27me3) to mediate transcriptional silencing. Loss-of-function SUZ12 alterations lead to PRC2 inactivation and are recurrent in malignant peripheral nerve sheath tumors (MPNST), where they are associated with epigenetic dysregulation.

Alterations observed in the corpus

  • Inactivating mutations and deletions in 33% of RT-MPNST vs 17% of sporadic MPNST, indicating enrichment in radiation-associated MPNST PMID:37350195.
  • SUZ12 undergoes homozygous and heterozygous deletions plus local genomic rearrangements producing aberrant transcripts in MPNST; mutually exclusive with EED loss; SUZ12 re-expression rescues H3K27me3 and inhibits growth PMID:25240281

Cancer types (linked)

  • MPNST – SUZ12 inactivation enriched in RT-MPNST (33%) compared to sporadic MPNST (17%); PRC2 complex component PMID:37350195.

Co-occurrence and mutual exclusivity

  • SUZ12 inactivation in MPNST co-occurs with NF1 inactivation (67% in RT-MPNST) and CDKN2A/CDKN2B deletions (92% in RT-MPNST) PMID:37350195.

Therapeutic relevance

  • Investigations on small molecular inhibitors of DNA methyltransferase (DNMT1) are ongoing in sporadic/NF1-related and RT-MPNSTs harboring PRC2-inactivating mutations such as SUZ12 loss PMID:37350195.

Open questions

  • Whether DNMT1 inhibitor efficacy differs between RT-MPNST and sporadic MPNST with PRC2 inactivation is not yet established PMID:37350195.

Sources

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